Vardenafil
Selleck Chemicals
SKU:E4803-5MG
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Vardenafil is an inhibitor of PDE used in studies of enzyme regulation. It is especially relevant in cardiovascular, metabolism, and neuroscience models, where defined compound exposure can be linked to catalytic activity, substrate turnover, and enzymatic regulation.
By inhibiting PDE, Vardenafil can be used to examine catalytic activity, substrate turnover, and enzymatic regulation. This target class is commonly examined through enzyme-activity assays, substrate-conversion studies, and mechanism profiling, together with downstream-response mapping. In cardiovascular, metabolism, and neuroscience models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.
Research Applications
- Target-focused assays involving PDE
- Concentration-response inhibition and target-dependence studies
- Enzyme-activity assays, substrate-conversion studies, and mechanism profiling
- Phenotypic profiling in cardiovascular, metabolism, and neuroscience models
Overall, Vardenafil is appropriate when a defined chemical perturbant is needed to connect PDE with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cardiovascular, metabolism, and neuroscience models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.
- Targets:
- PDE
- Target Class:
- Enzyme
- Research Area:
- Cardiovascular • Metabolism • Neuroscience
- CAS No.:
- 224785-90-4
- Molecular Weight:
- 488.60
- Formula:
- C₂₃H₃₂N₆O₄S
- SMILES:
- CCCc1nc(C)c2c(=O)nc(-c3cc(S(=O)(=O)N4CCN(CC)CC4)ccc3OCC)[nH]n12
- InChIKey:
- SECKRCOLJRRGGV-UHFFFAOYSA-N
- PubChem:
- 110634
- Storage Temperature:
- -20°C
For Research Use Only. Not intended for diagnostic or therapeutic use.
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