GSK-2881078

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Selleck Chemicals

S0276-5MG

€114,00 EUR
€114,00 EUR
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GSK-2881078 is a modulator of Androgen Receptor used in studies of Hormone Signaling. It is especially relevant in cancer and endocrinology models, where defined compound exposure can be linked to ligand-dependent transcriptional programs and endocrine regulation.

By modulating Androgen Receptor, GSK-2881078 can be used to examine ligand-dependent transcriptional programs and endocrine regulation. The nuclear receptor annotation adds relevance to reporter-gene, receptor-binding, and transcriptional assays, together with downstream-response mapping in the same experimental setting. In cancer and endocrinology models, these readouts can be combined with viability, reporter, localization, biochemical conversion, or morphology endpoints to refine experimental interpretation.

Research Applications

  • Target-focused assays involving Androgen Receptor
  • Pathway perturbation studies connected to Hormone Signaling
  • Context-dependent response profiling and mechanism comparison
  • Reporter-gene, receptor-binding, and transcriptional assays

Overall, GSK-2881078 is appropriate when a defined chemical perturbant is needed to connect Androgen Receptor with measurable biochemical, transcriptional, electrophysiological, imaging, or phenotypic readouts in cancer and endocrinology models. This profile is suited to mechanistic follow-up, comparative profiling, and assay optimization under defined exposure conditions.

Targets:
Androgen Receptor
Target Class:
Nuclear Receptor
Pathways:
Hormone Signaling
Research Area:
Cancer • Endocrinology
CAS No.:
1539314-06-1
Molecular Weight:
330.33
Formula:
C₁₄H₁₃F₃N₂O₂S
SMILES:
CC(CS(=O)(=O)C)N1C=CC2=C1C=CC(=C2C(F)(F)F)C#N
Storage Temperature:
-20°C

For Research Use Only. Not intended for diagnostic or therapeutic use.
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